SCHEMBL30133561

SCHEMBL30133561

CC(C)(C)OC(=O)N1CC(OC[C@H](NC(=O)OCC2c3ccccc3-c3ccccc32)C(=O)O)C1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 6/20 0.50
BACE1 P56817 1/20 0.49
MDM4 O15151 2/20 0.49
TP53 P04637 2/20 0.49
TNF P01375 1/20 0.45
TLR2 O60603 2/20 0.44
PRMT5 O14744 1/20 0.44
WDR77 Q9BQA1 1/20 0.44
CASP3 P42574 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30133512 0.93 BACE1 (0.49) MDM2BACE1MDM4TP53TNF
SCHEMBL22433653 0.91 BACE1 (0.52) MDM2BACE1MDM4TP53TNF
SCHEMBL24979705 0.89 BACE1 (0.47) MDM2BACE1MDM4TP53TNF
SCHEMBL22433654 0.89 BACE1 (0.47) MDM2BACE1MDM4TP53TNF
SCHEMBL31370469 0.84 MDM2 (0.49) MDM2BACE1MDM4TP53TLR2
SCHEMBL22433327 0.84 MDM2 (0.48) MDM2MDM4TP53TNFTLR2
SCHEMBL22579992 0.84 MDM2 (0.48) MDM2MDM4TP53TNFTLR2
SCHEMBL22552766 0.84 MDM2 (0.48) MDM2MDM4TP53TNFTLR2
SCHEMBL31688984 0.83 BACE1 (0.51) MDM2BACE1MDM4TP53TNF
SCHEMBL25267085 0.83 BACE1 (0.50) MDM2BACE1MDM4TP53CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12358951-B2 Cyclic peptide antibiotics GENENTECH, INC. (US) 2025-07-15 US disclosed
US-20230025834-A1 CYCLIC PEPTIDE ANTIBIOTICS GENENTECH, INC. (US) 2023-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230025834-A1 CYCLIC PEPTIDE ANTIBIOTICS NPPA, LNPEP, CLPP MDM2 2362/4885BACE1 404/4885MDM4 3536/4885
US-12358951-B2 Cyclic peptide antibiotics NPPA, LNPEP, CLPP MDM2 2362/4885BACE1 404/4885MDM4 3536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.