SCHEMBL30133894

SCHEMBL30133894

CON(C)C(=O)c1ccc2c(n1)C(C)(C)CO2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.33
DYRK1A Q13627 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
RARB P10826 2/20 0.33
RARG P13631 2/20 0.33
TRPM8 Q7Z2W7 1/20 0.31
MLYCD O95822 1/20 0.30
RARA P10276 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30899985 0.81 RARB (0.43) RARBRARGRARA
SCHEMBL30133991 0.81 RARB (0.43) RARBRARGRARA
SCHEMBL30133889 0.79 RARB (0.39) RARBRARGRARA
SCHEMBL30134106 0.79 RARB (0.36) RARBRARGRARA
SCHEMBL30540591 0.79 MAP3K14 (0.39) RARBRARGRARA
SCHEMBL8374791 0.68 KDM4E (0.45) CLK1DYRK1ADYRK1BTRPM8MLYCD
SCHEMBL30625585 0.68 RARB (0.45) RARBRARGRARA
SCHEMBL3739445 0.66 P2RX7 (0.49) CLK1DYRK1ADYRK1BTRPM8MLYCD
SCHEMBL31149391 0.66 NOTUM (0.35)
SCHEMBL25361140 0.65 RARA (0.46) RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125378-A2 Heterocyclic Compounds BEONE MEDICINES I GMBH (CH) 2026-05-07 US disclosed
EP-4658650-A1 HETEROCYCLIC COMPOUNDS Beone Medicines I GmbH (CH) 2025-12-10 EP disclosed
US-20250353846-A1 Heterocyclic Compounds BEONE MEDICINES I GMBH (CH) 2025-11-20 US disclosed
US-20240300951-A1 Pyrazolopyridinone Compounds BEIGENE LTD. (KY) 2024-09-12 US disclosed
US-20240270751-A1 Pyrazolopyridinone Compounds BEIGENE LTD. (KY) 2024-08-15 US disclosed
WO-2024160277-A1 HETEROCYCLIC COMPOUNDS BEIGENE, LTD. (KY) 2024-08-08 WO disclosed
EP-4380936-A1 PYRAZOLOPYRIDINONE COMPOUNDS BeiGene, Ltd. (KY) 2024-06-12 EP disclosed
WO-2023011456-A1 PYRAZOLOPYRIDINONE COMPOUNDS BEIGENE, LTD. (KY) 2023-02-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125378-A2 Heterocyclic Compounds NFATC1, CD4, MALT1 CLK1 4656/4885DYRK1A 4268/4885DYRK1B 4170/4885
US-20250353846-A1 Heterocyclic Compounds NFATC1, CD4, ACIN1 CLK1 3648/4885DYRK1A 4722/4885DYRK1B 4795/4885
US-20240300951-A1 Pyrazolopyridinone Compounds NFATC1, CD4, PBK CLK1 2511/4885DYRK1A 4397/4885DYRK1B 4467/4885
US-20240270751-A1 Pyrazolopyridinone Compounds NFATC1, CD4, PBK CLK1 2511/4885DYRK1A 4397/4885DYRK1B 4467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.