SCHEMBL30136007

SCHEMBL30136007

CCCCOC(=O)N1CC2(CCN(c3ncc(C4CCC(=O)NC4=O)cn3)CC2)C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 9/20 0.48
HSD17B10 Q99714 2/20 0.37
TSHR P16473 1/20 0.37
NPC1 O15118 1/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 1/20 0.36
DDB1 Q16531 7/20 0.35
GPR119 Q8TDV5 1/20 0.35
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ENPP2 Q13822 1/20 0.33
ATXN2 Q99700 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25035460 0.84 DDB1 (0.52) CRBNDDB1GPR119
SCHEMBL30475447 0.82 CRBN (0.41) CRBNHSD17B10TSHRKMT2ADDB1
SCHEMBL30135914 0.81 CRBN (0.48) CRBNHSD17B10TSHRNPC1POLB
SCHEMBL30135908 0.79 HSD17B10 (0.42) HSD17B10TSHRPOLBKMT2AGPR119
SCHEMBL30441826 0.79 CRBN (0.55) CRBNNPC1POLBKMT2ADDB1
SCHEMBL30135777 0.76 CRBN (0.48) CRBNHSD17B10TSHRNPC1POLB
SCHEMBL30135848 0.75 LMNA (0.39) HSD17B10TSHRPOLBKMT2AGPR119
SCHEMBL25035459 0.74 CRBN (0.44) CRBNHSD17B10TSHRPOLBDDB1
SCHEMBL25825240 0.73 CRBN (0.41) CRBNPOLBDDB1
SCHEMBL30135799 0.72 CRBN (0.51) CRBNNPC1DDB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157849-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2023-04-05 EP disclosed
WO-2023017446-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed
WO-2023018238-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-02-16 WO disclosed