SCHEMBL30137270

SCHEMBL30137270

Cn1nc(NC(=O)OCc2ccccc2)c2ccc(N3CC4(CCNCC4)C3)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
ROCK2 O75116 1/20 0.39
MAPK1 P28482 3/20 0.39
USP2 O75604 2/20 0.39
ALDH1A1 P00352 2/20 0.39
TP53 P04637 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HIF1A Q16665 1/20 0.39
TSHR P16473 2/20 0.38
LRRK2 Q5S007 2/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
FLT1 P17948 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
BTK Q06187 1/20 0.36
FAAH O00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27242958 0.89 ITGB3 (0.41) SMN1; SMN2MAPK1USP2ALDH1A1CYP1A2
SCHEMBL30990853 0.85 HSD17B10 (0.41) SMN1; SMN2MAPK1USP2ALDH1A1CYP1A2
SCHEMBL30137486 0.76 SMN1; SMN2 (0.50) SMN1; SMN2ROCK2ALDH1A1MGLL
SCHEMBL8589894 0.70 HTR3A (0.50) SMN1; SMN2ALDH1A1KDR
SCHEMBL7711512 0.68 ENPP2 (0.54) SMN1; SMN2MAPK1ALDH1A1CYP1A2HIF1A
SCHEMBL25026452 0.67 KHK (0.34) KHKSMN1; SMN2MAPK1USP2ALDH1A1
SCHEMBL8305123 0.66 HTR3A (0.54) SMN1; SMN2TSHRKDRFLT3
SCHEMBL31635906 0.65 TMEM97 (0.55) SMN1; SMN2
SCHEMBL25026459 0.65 DDB1 (0.65) KHKSMN1; SMN2MAPK1USP2ALDH1A1
SCHEMBL27953763 0.64 POLB (0.54) SMN1; SMN2ROCK2USP2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023016518-A1 HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF 四川海思科制药有限公司 2023-02-16 WO disclosed