SCHEMBL30149233

SCHEMBL30149233

CC(C)(C)OC(=O)C(Br)c1cncc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.37
ADORA2A P29274 14/20 0.36
ADORA1 P30542 3/20 0.36
ADORA3 P0DMS8 3/20 0.36
ADORA2B P29275 13/20 0.36
APP P05067 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP3A5 P20815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27395438 0.76 APP (0.41) APP
SCHEMBL25908715 0.76 ADORA2A (0.39) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9462640 0.75 RAB9A (0.43) CYP3A4CYP3A5
SCHEMBL25281119 0.71 APP (0.45) APP
SCHEMBL30437614 0.70 HCAR2 (0.55) HCAR2CYP3A4
SCHEMBL355454 0.69 CES2 (0.53)
SCHEMBL25232209 0.69 ADORA2A (0.42) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL22608911 0.69 ADORA2A (0.37) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL31205660 0.69 ADORA2A (0.42) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL25261485 0.69 ADORA2A (0.42) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022221686-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2022-10-20 WO disclosed