SCHEMBL3016592

SCHEMBL3016592

Cc1cc(C)c(S(=O)(=O)C2CCN(c3nc(Cc4ccc(Cl)c(Cl)c4)cs3)CC2)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.42
LMNA P02545 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
AR P10275 1/20 0.36
FPR2 P25090 1/20 0.36
PROKR1 Q8TCW9 1/20 0.36
DNM1L O00429 7/20 0.34
APAF1 O14727 1/20 0.34
PKM P14618 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3005486 0.92 PROKR1 (0.38) EPHX2LMNAL3MBTL1FPR2PROKR1
SCHEMBL3012456 0.92 SOS1 (0.38) EPHX2LMNADNM1L
SCHEMBL3018899 0.92 LMNA (0.39) EPHX2LMNAL3MBTL1ARFPR2
SCHEMBL3007167 0.91 EPHX2 (0.39) EPHX2LMNADNM1LMEN1KMT2A
SCHEMBL3016255 0.90 DNM1L (0.35) ARDNM1LMEN1KMT2A
SCHEMBL3016483 0.89 SMN1; SMN2 (0.39) ARDNM1LMEN1KMT2A
SCHEMBL3018927 0.89 DNM1L (0.36) EPHX2DNM1LMEN1KMT2A
SCHEMBL3012727 0.88 ALDH1A1 (0.40) LMNAL3MBTL1ARDNM1LKMT2A
SCHEMBL3011125 0.88 DNM1L (0.35) LMNADNM1LMEN1KMT2A
SCHEMBL3002261 0.87 DNM1L (0.38) DNM1LMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8722681-B2 N-sulfonyl thiazolylpiperazine derivatives and related N-sulfonyl heterocyclic derivatives for the treatment of neuro degenerative diseases NV REMYND (BE) 2014-05-13 US disclosed
US-20100197703-A1 N-SULFONYL THIAZOLYLPIPERAZINE DERIVATIVES AND RELATED N-SULFONYL HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF NEURO DEGENERATIVE DISEASES NV REMYND (BE) 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197703-A1 N-SULFONYL THIAZOLYLPIPERAZINE DERIVATIVES AND RELATED N-SULFONYL HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF NEURO DEGENERATIVE DISEASES SMN1; SMN2, HTT, SNCA EPHX2 4409/4885LMNA 80/4885L3MBTL1 1847/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.