SCHEMBL30178342

SCHEMBL30178342

COCOCCCn1c(=O)c(Br)cn(CC(=O)O)c1=O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.36
ADORA2B P29275 6/20 0.33
ADORA2A P29274 5/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
ALDH1A1 P00352 4/20 0.32
LMNA P02545 1/20 0.32
TNF P01375 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17870788 0.93 CDK9 (0.37) CDK9ADORA2BADORA2APDE4APDE4B
SCHEMBL17870758 0.85 ALDH1A1 (0.41) CDK9ADORA2BADORA2APDE4APDE4B
SCHEMBL28651571 0.82 CDK9 (0.39) CDK9ALDH1A1TNFKDM4EMAPT
SCHEMBL17870821 0.78 CDK9 (0.42) CDK9ADORA2BADORA2APDE4APDE4B
SCHEMBL17870748 0.78 CDK9 (0.39) CDK9ADORA2BADORA2APDE4APDE4B
SCHEMBL19873765 0.76 ALDH1A1 (0.38) CDK9ADORA2BALDH1A1TNFMAPT
SCHEMBL17870770 0.76 CDK9 (0.41) CDK9ADORA2BPDE4APDE4BPDE4C
SCHEMBL21900263 0.75 CDK9 (0.44) CDK9ADORA2BALDH1A1LMNAKDM4E
SCHEMBL17870749 0.75 CDK9 (0.40) CDK9ADORA2BALDH1A1LMNAKDM4E
SCHEMBL17870790 0.74 CDK9 (0.38) CDK9ALDH1A1LMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3708566-B1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RES & DEV (FR) 2023-02-08 EP disclosed