SCHEMBL30178741

SCHEMBL30178741

CSC(C)Cn1c(=O)c(Br)cn(CC(=O)O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 1/20 0.39
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.32
GRIA1 P42261 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA4 P48058 1/20 0.32
GRIK5 Q16478 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21900226 0.86 CDK9 (0.41) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL21900263 0.79 CDK9 (0.44) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL17870749 0.78 CDK9 (0.40) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL17870748 0.76 CDK9 (0.39) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL17870821 0.76 CDK9 (0.42) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL19873909 0.76 ALDH1A1 (0.39) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL21900243 0.76 ALDH1A1 (0.35) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL21900244 0.76 ALDH1A1 (0.35) CDK9ALDH1A1KDM4EPOLBMAPT
SCHEMBL30178325 0.75 GNRHR (0.46)
SCHEMBL17870770 0.74 CDK9 (0.41) CDK9ALDH1A1KDM4EPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3708566-B1 NOVEL HETEROCYCLIC COMPOUNDS AND THE USE THEREOF IN MEDICINE AND IN COSMETICS GALDERMA RES & DEV (FR) 2023-02-08 EP disclosed