SCHEMBL30185581

SCHEMBL30185581

O=C1NCC(C(F)(F)F)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP3 Q9Y6F1 1/20 0.50
PARP1 P09874 4/20 0.43
PARP2 Q9UGN5 1/20 0.43
HTR2A P28223 4/20 0.42
HTR2C P28335 4/20 0.42
HTR2B P41595 4/20 0.42
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
HSD17B10 Q99714 1/20 0.38
PARP10 Q53GL7 2/20 0.38
PARP11 Q9NR21 2/20 0.38
PDPK1 O15530 1/20 0.38
TNKS2 Q9H2K2 2/20 0.36
GSK3B P49841 1/20 0.34
CYP1A2 P05177 1/20 0.34
HTT P42858 1/20 0.33
NCOA1 Q15788 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Boric Acid SCHEMBL29099586 0.94 PARP3 (0.49) PARP3PARP1PARP2HTR2AHTR2C
SCHEMBL8931375 0.84 PARP3 (0.49) PARP3PARP1PARP2HTR2AHTR2C
SCHEMBL31412980 0.77 PARP10 (0.44) PARP3PARP1HTR2AHTR2CHTR2B
SCHEMBL26510292 0.77 PARP10 (0.44) PARP3PARP1HTR2AHTR2CHTR2B
SCHEMBL26121467 0.77 TDP2 (0.37) PARP3PARP1PARP2PARP10PARP11
SCHEMBL25758208 0.76 HTR2C (0.33) PARP1PARP2HTR2CTNKS2
SCHEMBL29458430 0.74 PARP3 (0.43) PARP3PARP1PARP2HTR2AHTR2C
SCHEMBL6635520 0.74 PARP3 (0.53) PARP3PARP1HTR2AHTR2CHTR2B
SCHEMBL21187107 0.74 PARP3 (0.53) PARP3PARP1PARP2HTR2AHTR2C
SCHEMBL12220005 0.74 PARP3 (0.53) PARP3PARP1HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-B PI3K alpha inhibitor with double-ring structure, and preparation method and application thereof 生物岛实验室 2025-03-28 CN disclosed
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed