SCHEMBL21187107

SCHEMBL21187107

O=C1NCC(I)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP3 Q9Y6F1 2/20 0.53
HTR2A P28223 3/20 0.45
HTR2C P28335 3/20 0.45
HTR2B P41595 3/20 0.45
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
PARP1 P09874 5/20 0.41
PARP10 Q53GL7 2/20 0.40
PARP11 Q9NR21 2/20 0.40
PDPK1 O15530 1/20 0.40
GSK3B P49841 1/20 0.37
HSD17B10 Q99714 2/20 0.37
PARP2 Q9UGN5 1/20 0.35
PIM1 P11309 1/20 0.34
CSNK1A1 P48729 1/20 0.34
CDK5 Q00535 1/20 0.34
ROCK1 Q13464 1/20 0.34
DYRK1A Q13627 1/20 0.34
LRRK2 Q5S007 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635520 0.77 PARP3 (0.53) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL11750196 0.77 PARP3 (0.61) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL12220005 0.77 PARP3 (0.53) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL30185581 0.74 PARP3 (0.50) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL1315337 0.74 PARP3 (0.62) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL8931375 0.73 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL21187169 0.73 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL29594704 0.73 PARP3 (0.56) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL21187216 0.73 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12
SCHEMBL29458586 0.73 PARP3 (0.49) PARP3HTR2AHTR2CHTR2BCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed