SCHEMBL30185583

SCHEMBL30185583

O=C(O)CC(c1cccc(Br)c1)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.47
MGAM O43451 1/20 0.41
GAA P10253 1/20 0.41
SI P14410 1/20 0.41
MGAM2 Q2M2H8 1/20 0.41
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
FFAR1 O14842 1/20 0.40
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
ALDH1A1 P00352 1/20 0.38
SLC6A9 P48067 2/20 0.38
CYP26A1 O43174 1/20 0.38
IDO1 P14902 2/20 0.37
TDO2 P48775 1/20 0.37
GABBR2 O75899 1/20 0.37
GABBR1 Q9UBS5 1/20 0.37
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29099531 1.00 CTSA (0.47) CTSAMGAMGAASIMGAM2
SCHEMBL3658761 0.83 KYNU (0.44) GAASMN1; SMN2FFAR1IDO1GABBR2
SCHEMBL3660011 0.83 KYNU (0.44) GAASMN1; SMN2FFAR1IDO1GABBR2
SCHEMBL29099504 0.82 KCNA5 (0.47) CTSAALDH1A1
SCHEMBL30185560 0.82 KCNA5 (0.47) CTSAALDH1A1
SCHEMBL19817286 0.81 GABBR2 (0.48) FFAR1FNTAFNTBGABBR2GABBR1
SCHEMBL3053473 0.81 GABBR2 (0.48) FFAR1FNTAFNTBGABBR2GABBR1
SCHEMBL23125123 0.81 ACP3 (0.50) CTSASMN1; SMN2ALDH1A1SLC6A9IDO1
SCHEMBL1932025 0.81 CPN1 (0.49) SMN1; SMN2FFAR1IDO1GABBR2GABBR1
SCHEMBL7141329 0.78 FNTA (0.53) CTSAMGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024125464-A1 TETRAHYDROISOQUINOLIN-ONE DERIVATIVES, PREPARATION METHODS AND MEDICINAL USES THEREOF JIANGSU HANSOH PHARMACEUTICAL GROUP CO., LTD. (CN) 2024-06-20 WO disclosed
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed