SCHEMBL30186173

SCHEMBL30186173

Cc1sc(Nc2ccc(Cl)cc2F)nc1C(=O)N1CCC[C@H](C)[C@@H]1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPC3 Q13507 10/20 1.00
TRPC6 Q9Y210 10/20 1.00
TRPA1 O75762 2/20 1.00
CACNA1C Q13936 2/20 1.00
SCN5A Q14524 2/20 1.00
TRPV1 Q8NER1 2/20 1.00
TRPV4 Q9HBA0 2/20 1.00
HCRTR1 O43613 10/20 0.41
HCRTR2 O43614 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26459111 1.00 TRPC3 (1.00) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL798463 1.00 TRPC3 (1.00) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL26458205 0.91 TRPC3 (0.83) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL26458213 0.91 TRPC3 (0.83) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL789038 0.87 TRPC3 (0.77) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL790188 0.84 TRPC3 (0.72) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL806600 0.84 TRPC3 (1.00) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL26459144 0.84 TRPC3 (0.72) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL790044 0.83 TRPC3 (0.71) TRPC3TRPC6TRPA1CACNA1CSCN5A
SCHEMBL806708 0.81 TRPC3 (0.68) TRPC3TRPC6TRPA1CACNA1CSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4103245-B1 ADMINISTRATION OF CALCIUM CHANNEL TRPC6 INHIBITORS USING BALLOONS, STENTS OR OTHER MEDICAL DEVICES KLINIKUM DER TECHNISCHEN UNIV MUENCHEN TUM KLINIKUM (DE) 2026-04-01 EP disclosed
CN-112204017-B Benzisoxazole compounds 国立大学法人大阪大学 2024-08-20 CN disclosed
US-11976062-B2 Benzisoxazole compound OSAKA UNIVERSITY (JP) 2024-05-07 US disclosed
EP-3789383-B9 INHIBITORS OF THE TRPC3 OR TRPC6 CHANNEL UNIV OSAKA (JP) 2024-02-28 EP disclosed
EP-3789383-B1 INHIBITORS OF THE TRPC3 OR TRPC6 CHANNEL UNIV OSAKA (JP) 2023-11-29 EP disclosed
US-20230137816-A1 ADMINISTRATION OF CALCIUM CHANNEL TRPC6 INHIBITORS USING BALLOONS, STENTS OR OTHER MEDICAL DEVICES DEUTSCHES HERZZENTRUM MUENCHEN DES FREISTAATES BAYERN (DE) 2023-05-04 US disclosed
US-20230114195-A1 BENZISOXAZOLE COMPOUND KYOTO UNIVERSITY (JP) 2023-04-13 US disclosed
US-11548882-B2 Benzisoxazole compound OSAKA UNIVERSITY (JP) 2023-01-10 US disclosed
EP-4103245-A1 ADMINISTRATION OF CALCIUM CHANNEL TRPC6 INHIBITORS USING BALLOONS, STENTS OR OTHER MEDICAL DEVICES Klinikum rechts der Isar der Technischen Universität München (DE) 2022-12-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230137816-A1 ADMINISTRATION OF CALCIUM CHANNEL TRPC6 INHIBITORS USING BALLOONS, STENTS OR OTHER MEDICAL DEVICES TRPC6, TRPC1, ORAI1 TRPC3 6/4885TRPC6 1/4885TRPA1 26/4885
US-11976062-B2 Benzisoxazole compound CBR1, CYP2S1, CYP2E1 TRPC3 2975/4885TRPC6 3601/4885TRPA1 1638/4885
US-11548882-B2 Benzisoxazole compound CBR1, CYP2S1, CYP2E1 TRPC3 3014/4885TRPC6 3644/4885TRPA1 1697/4885
US-20230114195-A1 BENZISOXAZOLE COMPOUND CBR1, CYP2S1, CYP2E1 TRPC3 2830/4885TRPC6 3541/4885TRPA1 1702/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.