SCHEMBL30189323

SCHEMBL30189323

C=C(C(=O)OC)C(O)c1cc(C(F)F)ccn1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.34
AAK1 Q2M2I8 4/20 0.32
RIOK2 Q9BVS4 1/20 0.30
SYK P43405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29301526 0.82 TP53 (0.37) RIOK2
SCHEMBL31613977 0.81 KDM4C (0.39) SMARCA2
SCHEMBL27972604 0.81 KDM4E (0.38)
SCHEMBL30189285 0.81 P2RX7 (0.33)
SCHEMBL22615150 0.81 KDM4C (0.39) SMARCA2
SCHEMBL27972528 0.77 EGFR (0.42) RIOK2
SCHEMBL24586223 0.76 CYP3A4 (0.41)
SCHEMBL14915338 0.76 CYP3A4 (0.41)
SCHEMBL29925482 0.76 CYP3A4 (0.41)
SCHEMBL22615180 0.70 APLNR (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4149945-A1 SUBSTITUTED TRICYCLIC AMIDES, ANALOGUES THEREOF, AND METHODS USING SAME Arbutus Biopharma Corporation (CA) 2023-03-22 EP disclosed