SCHEMBL30189933

SCHEMBL30189933

COCc1cnc2c(Br)cc(Cl)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 1/20 0.33
CA2 P00918 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19783603 1.00 S1PR4 (0.33) S1PR4CA2CYP11B1CYP11B2ALDH1A1
SCHEMBL30189953 0.83 CCR1 (0.34) CA2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL19782862 0.83 CCR1 (0.34) CA2CYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL19783747 0.83 PARP1 (0.39)
SCHEMBL30189663 0.79 ENPP2 (0.33) CYP11B1CYP11B2
SCHEMBL21395879 0.79 ENPP2 (0.33) CYP11B1CYP11B2
SCHEMBL19776056 0.76 ALDH1A1 (0.35) ALDH1A1MAPTSMN1; SMN2
SCHEMBL19783099 0.76
SCHEMBL19776449 0.76 S1PR4 (0.39) S1PR4ALDH1A1LMNAMAPTHPGD
SCHEMBL29481826 0.76 S1PR4 (0.39) S1PR4ALDH1A1LMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396469-A Inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-12 CN disclosed
CN-109689647-B Bicyclic heteroaryl substituted compounds 百时美施贵宝公司 2023-01-20 CN disclosed