SCHEMBL30201250

SCHEMBL30201250

O=C(O)Cc1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
FFAR4 Q5NUL3 1/20 0.47
MRGPRX4 Q96LA9 3/20 0.47
RXRA P19793 2/20 0.47
RXRB P28702 2/20 0.47
RXRG P48443 2/20 0.47
PPARD Q03181 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNJ5 P48544 1/20 0.46
KCNJ3 P48549 1/20 0.46
PSEN1 P49768 1/20 0.45
PSEN2 P49810 1/20 0.45
APH1B Q8WW43 1/20 0.45
NCSTN Q92542 1/20 0.45
APH1A Q96BI3 1/20 0.45
PSENEN Q9NZ42 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1775542 1.00 ALDH1A1 (0.52) ALDH1A1FFAR4MRGPRX4RXRARXRB
SCHEMBL29718989 0.86 RXRA (0.50) ALDH1A1MRGPRX4RXRARXRBRXRG
SCHEMBL838070 0.86 RXRA (0.50) ALDH1A1MRGPRX4RXRARXRBRXRG
SCHEMBL14263413 0.85 ALDH1A1 (0.45) ALDH1A1FFAR4MRGPRX4MEN1KMT2A
SCHEMBL30591389 0.85 ALDH1A1 (0.48) ALDH1A1FFAR4MRGPRX4MEN1KMT2A
SCHEMBL31750436 0.83 FFAR1 (0.54) ALDH1A1FFAR4MEN1KMT2AKCNJ5
SCHEMBL31204321 0.83 ALDH1A1 (0.44) ALDH1A1FFAR4MRGPRX4MEN1KMT2A
Trifluoroacetic Acid SCHEMBL5769358 0.82 FFAR1 (0.47) ALDH1A1FFAR4MRGPRX4RXRARXRB
Hydrochloric Acid SCHEMBL34474962 0.82 FFAR1 (0.53) ALDH1A1FFAR4MEN1KMT2AKCNJ5
Trifluoroacetic Acid SCHEMBL34475312 0.81 FFAR1 (0.52) ALDH1A1FFAR4MEN1KMT2AKCNJ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023028056-A1 3-AMINO PIPERIDYL SODIUM CHANNEL INHIBITORS GENENTECH, INC. (US) 2023-03-02 WO disclosed