SCHEMBL30201440

SCHEMBL30201440

O=C(O)c1ccc2cc(C(F)(F)F)[nH]c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.55
CASP3 P42574 1/20 0.54
SENP8 Q96LD8 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
SENP6 Q9GZR1 1/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
HPGD P15428 1/20 0.53
ENPP2 Q13822 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CHEK2 O96017 2/20 0.47
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
HSP90AA1 P07900 1/20 0.44
ESR2 Q92731 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ITK Q08881 1/20 0.44
NOTUM Q6P988 1/20 0.44
PTPN1 P18031 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24950452 1.00 SMN1; SMN2 (0.55) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL28128641 0.85 CHEK2 (0.43) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL3922415 0.83 CASP3 (0.54) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL30445643 0.75 HSD17B10 (0.61) CASP3SENP8SENP7SENP6KDM4E
SCHEMBL31721323 0.75 CASP3 (0.60) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL69851 0.75 HSD17B10 (0.61) CASP3SENP8SENP7SENP6KDM4E
SCHEMBL24950978 0.74 TAS1R3 (0.52) KDM4EALDH1A1
SCHEMBL19476290 0.74 CASP3 (0.58) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL233323 0.74 CASP3 (0.58) SMN1; SMN2CASP3SENP8SENP7SENP6
SCHEMBL5868213 0.74 CASP3 (0.58) SMN1; SMN2CASP3SENP8SENP7SENP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117729914-A Serotonin 5-HT2B inhibiting compounds 硕腾服务有限责任公司 2024-03-19 CN disclosed
WO-2023009330-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC (US) 2023-02-02 WO disclosed