SCHEMBL30205259

SCHEMBL30205259

COc1ccc(-c2c(S(N)(=O)=O)ccc(N3CCN(Cc4cccc([N+](=O)[O-])c4)CC3)c2[N+](=O)[O-])cn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYD88 Q99836 2/20 0.59
ALDH1A1 P00352 7/20 0.44
KDM4E B2RXH2 4/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
GFER P55789 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 3/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPK1 P28482 3/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205261 0.91 MYD88 (0.48) MYD88ALDH1A1KDM4ELMNACYP3A4
SCHEMBL30205266 0.83 CA1 (0.45) MYD88TDP1MEN1KMT2APOLB
SCHEMBL28954767 0.74 MYD88 (1.00) MYD88ALDH1A1KDM4ETDP1MEN1
SCHEMBL30585268 0.73 MYD88 (0.55) MYD88ALDH1A1KDM4ETDP1MEN1
SCHEMBL28954834 0.71 MYD88 (0.64) MYD88ALDH1A1MEN1GAAKMT2A
SCHEMBL29078406 0.70 MYD88 (0.68) MYD88ALDH1A1KDM4ETDP1MEN1
SCHEMBL30585272 0.69 ALDH1A1 (0.55) MYD88ALDH1A1KDM4ETDP1MEN1
SCHEMBL29078389 0.68 MYD88 (0.60) MYD88ALDH1A1KDM4ETDP1MEN1
SCHEMBL15800712 0.67 ALDH1A1 (0.78) ALDH1A1KDM4ETDP1MEN1GAA
SCHEMBL6858096 0.65 MEN1 (0.65) ALDH1A1KDM4ETDP1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710251-A Myeloid differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2023-02-24 CN disclosed