SCHEMBL30205261

SCHEMBL30205261

COc1ccc(-c2c(S(N)(=O)=O)ccc(N3CCN(Cc4ccc([N+](=O)[O-])cc4)CC3)c2[N+](=O)[O-])cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYD88 Q99836 1/20 0.48
ALDH1A1 P00352 5/20 0.40
LMNA P02545 1/20 0.40
CASP1 P29466 1/20 0.40
CASP4 P49662 1/20 0.40
CASP5 P51878 1/20 0.40
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABCB1 P08183 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
POLB P06746 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
NPBWR1 P48145 1/20 0.38
MCHR1 Q99705 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205259 0.91 MYD88 (0.59) MYD88ALDH1A1LMNAMAPTCYP3A4
SCHEMBL30205266 0.83 CA1 (0.45) MYD88MAPTPOLBCA12CA1
SCHEMBL28954891 0.72 MYD88 (0.85) MYD88ALDH1A1LMNAMAPTHTT
SCHEMBL30585285 0.72 ALDH1A1 (0.46) MYD88ALDH1A1LMNAHTTABCC1
SCHEMBL28954834 0.69 MYD88 (0.64) MYD88ALDH1A1LMNAMAPTHTT
SCHEMBL29078361 0.69 MYD88 (0.55) MYD88ALDH1A1LMNAHTTPOLB
SCHEMBL209309 0.68 TRPV6 (0.41) MYD88ALDH1A1MAPTNPBWR1MCHR1
SCHEMBL30585270 0.67 ALDH1A1 (0.46) ALDH1A1LMNAHTTABCB1ABCG2
SCHEMBL29078394 0.66 MEN1 (0.60) MYD88ALDH1A1LMNAMAPTHTT
SCHEMBL11556531 0.66 MAPK1 (0.69) ALDH1A1LMNAMAPTABCC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710251-A Myeloid differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2023-02-24 CN disclosed