SCHEMBL30212975

SCHEMBL30212975

Nc1cccc(-c2c[nH]nn2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.50
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 3/20 0.47
KDM4E B2RXH2 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 2/20 0.47
KMT2A Q03164 2/20 0.47
MAOA P21397 1/20 0.45
CHEK1 O14757 1/20 0.45
TSHR P16473 1/20 0.44
RECQL P46063 1/20 0.44
GLA P06280 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MECP2 P51608 1/20 0.43
MAP4K4 O95819 2/20 0.43
ENPP2 Q13822 1/20 0.42
KIT P10721 2/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4313886 1.00 METAP2 (0.50) METAP2ALDH1A1MEN1KDM4ELMNA
SCHEMBL1646236 0.86 GP6 (0.37) METAP2ALDH1A1MEN1KMT2ACHEK1
SCHEMBL4831837 0.78 HSD17B1 (0.53) METAP2
SCHEMBL670668 0.78 IDO1 (0.50) METAP2ALDH1A1MEN1KDM4EMAPT
SCHEMBL5613019 0.78 METAP2 (0.50) METAP2
SCHEMBL13896466 0.78 IDO1 (0.50) MEN1KDM4ELMNAMAPTKMT2A
SCHEMBL7520387 0.78 AKT1 (0.31)
SCHEMBL917247 0.78 IDO1 (0.46)
SCHEMBL29899236 0.78 IDO1 (0.50) MEN1KDM4ELMNAMAPTKMT2A
SCHEMBL29746032 0.78 IDO1 (0.50) METAP2ALDH1A1MEN1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115697974-A Imidazole 3-oxide derivative based ACSS2 inhibitors and methods of use thereof 美特波米德有限公司 2023-02-03 CN disclosed