SCHEMBL30219271

SCHEMBL30219271

CSc1cc(C(N)=O)ccc1C

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AR P10275 14/20 0.50
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
PARP1 P09874 1/20 0.46
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL858842 0.85 TAS1R3 (0.55) ARTAS1R3TAS1R1PARP1
SCHEMBL701970 0.82 TAS1R3 (0.50) ARTAS1R3TAS1R1MAPTTDP1
SCHEMBL9548004 0.82 TAS1R3 (0.50) TAS1R3TAS1R1MAPTTDP1
SCHEMBL8606616 0.81 TAS1R3 (0.49) ARTAS1R3TAS1R1MAPTTDP1
SCHEMBL15855901 0.78 AR (0.48) ARPARP1TDP1
SCHEMBL21374189 0.78 ALDH1A1 (0.57) TAS1R3TAS1R1MAPTTDP1
SCHEMBL13495890 0.78 PARP1 (0.40) ARPARP1MAPTTDP1
SCHEMBL1002832 0.77 PRSS1 (0.61) PARP1MAPTTDP1
SCHEMBL29503140 0.77 PRSS1 (0.61) PARP1MAPTTDP1
SCHEMBL858817 0.77 AR (0.57) ARPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN claimed
CN-116715625-A Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-09-08 CN disclosed
CN-111601790-B Heteroaryl compounds as protein kinase inhibitors 福建海西新药创制股份有限公司 2023-03-31 CN disclosed