SCHEMBL9548004

SCHEMBL9548004

CSc1cc(C(C)=O)ccc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.50
TAS1R1 Q7RTX1 2/20 0.50
CRHR1 P34998 1/20 0.48
CYP2A6 P11509 1/20 0.44
ALDH1A1 P00352 3/20 0.43
HPGD P15428 4/20 0.42
LMNA P02545 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
RAB9A P51151 5/20 0.41
MAPT P10636 5/20 0.41
NPC1 O15118 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HSD17B1 P14061 1/20 0.40
PKM P14618 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
PRKCI P41743 1/20 0.38
S100A4 P26447 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK1 P28482 1/20 0.37
STAT3 P40763 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10361232 0.84 TAS1R3 (0.57) TAS1R3TAS1R1CRHR1CYP2A6ALDH1A1
SCHEMBL701970 0.84 TAS1R3 (0.50) TAS1R3TAS1R1ALDH1A1L3MBTL1MAPT
SCHEMBL30219271 0.82 AR (0.50) TAS1R3TAS1R1MAPTTDP1
SCHEMBL8606616 0.82 TAS1R3 (0.49) TAS1R3TAS1R1CRHR1ALDH1A1HPGD
SCHEMBL1545562 0.80 PKM (0.52) CRHR1CYP2A6ALDH1A1HPGDLMNA
SCHEMBL21374189 0.79 ALDH1A1 (0.57) TAS1R3TAS1R1ALDH1A1HPGDLMNA
SCHEMBL9548058 0.78 GSK3B (0.52) TAS1R3TAS1R1L3MBTL1KMT2A
SCHEMBL29787835 0.76 SMN1; SMN2 (0.57) CYP2A6ALDH1A1HPGDLMNARAB9A
SCHEMBL110321 0.76 SMN1; SMN2 (0.57) CYP2A6ALDH1A1HPGDLMNARAB9A
SCHEMBL10804813 0.76 ALDH1A1 (0.51) ALDH1A1HPGDLMNAL3MBTL1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198587-A Adrenergic Blocking Agents, Hypotensive Agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1993-03-30 US disclosed
US-5063246-A Hypotensive YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-11-05 US disclosed
US-4880841-A ADRENERGIC BLOCKING AGENTS, HYPOTENSIVE AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1989-11-14 US disclosed