SCHEMBL3022148

SCHEMBL3022148

CCCc1ccc(Cc2csc(N3CCC(S(=O)(=O)c4ccc(Cl)c(Cl)c4)CC3)n2)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
THRB P10828 1/20 0.35
ADAMTS5 Q9UNA0 2/20 0.33
ERBB2 P04626 2/20 0.33
EPHA2 P29317 2/20 0.33
KDR P35968 2/20 0.33
EPHB4 P54760 2/20 0.33
AR P10275 1/20 0.33
KIT P10721 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
AOC3 Q16853 1/20 0.33
NFE2L2 Q16236 1/20 0.33
DNM1L O00429 1/20 0.33
KDM2B Q8NHM5 1/20 0.32
HTR7 P34969 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3010484 0.93 THRB (0.42) LMNAL3MBTL1THRBERBB2EPHA2
SCHEMBL3016262 0.92 HTR2A (0.36) L3MBTL1ADAMTS5KITHTR2AHTR2C
SCHEMBL3016660 0.91 GBA1 (0.38) LMNAL3MBTL1THRBARDNM1L
SCHEMBL3017117 0.91 MAPT (0.38) LMNAL3MBTL1ARHTR2AHTR2C
SCHEMBL3013801 0.91 L3MBTL1 (0.39) LMNAL3MBTL1THRBERBB2EPHA2
SCHEMBL3001978 0.90 VCAM1 (0.39) LMNA
SCHEMBL3012962 0.90 AOC3 (0.34) LMNAADAMTS5KITHTR2AHTR2C
SCHEMBL3016706 0.90 MAPT (0.37) LMNAHTR2AHTR2C
SCHEMBL3015155 0.89 HTR2A (0.41) LMNAL3MBTL1ARHTR2AHTR2C
SCHEMBL3011356 0.89 MAPT (0.39) LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8722681-B2 N-sulfonyl thiazolylpiperazine derivatives and related N-sulfonyl heterocyclic derivatives for the treatment of neuro degenerative diseases NV REMYND (BE) 2014-05-13 US disclosed
US-20100197703-A1 N-SULFONYL THIAZOLYLPIPERAZINE DERIVATIVES AND RELATED N-SULFONYL HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF NEURO DEGENERATIVE DISEASES NV REMYND (BE) 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197703-A1 N-SULFONYL THIAZOLYLPIPERAZINE DERIVATIVES AND RELATED N-SULFONYL HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF NEURO DEGENERATIVE DISEASES SMN1; SMN2, HTT, SNCA LMNA 80/4885L3MBTL1 1847/4885THRB 2628/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.