SCHEMBL30234729

SCHEMBL30234729

Fc1cc(NCC(F)(F)F)c(Br)c(OCc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.41
MAPK14 Q16539 6/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
LMNA P02545 3/20 0.38
LRRK2 Q5S007 1/20 0.38
PTGER1 P34995 1/20 0.36
CCR5 P51681 2/20 0.36
MAPT P10636 2/20 0.36
FFAR1 O14842 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PPIA P62937 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23883903 1.00 KDM1A (0.41) KDM1AMAPK14L3MBTL1LMNALRRK2
SCHEMBL30335270 0.78 CTSV (0.44) KDM1AMAPK14L3MBTL1LMNALRRK2
SCHEMBL23883904 0.78 CTSV (0.44) KDM1AMAPK14L3MBTL1LMNALRRK2
SCHEMBL26133457 0.77 MRGPRX4 (0.48) KDM1AMAPK14L3MBTL1PTGER1MAPT
SCHEMBL4540283 0.76 KDM1A (0.56) KDM1AMAPK14L3MBTL1LMNALRRK2
SCHEMBL23883871 0.76 KDM1A (0.49) KDM1AMAPK14L3MBTL1LRRK2PTGER1
SCHEMBL30335518 0.76 KDM1A (0.49) KDM1AMAPK14L3MBTL1LRRK2PTGER1
SCHEMBL23899806 0.74 HTR1A (0.43) KDM1AMAPK14L3MBTL1LMNALRRK2
SCHEMBL23899537 0.74 KDM1A (0.50) KDM1AMAPK14L3MBTL1LRRK2PTGER1
SCHEMBL30234551 0.72 CTSV (0.45) KDM1AMAPK14L3MBTL1LRRK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4132908-A1 INDOLE DERIVATIVES AS ALPHA-1 -ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1 -ANTITRYPSIN DEFICIENCY (AATD) Vertex Pharmaceuticals Incorporated (US) 2023-02-15 EP disclosed