SCHEMBL3025015

SCHEMBL3025015

CNC(=O)c1cccc(-c2ccn3c(Br)cnc3c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 3/20 0.49
FGFR1 P11362 2/20 0.49
FYN P06241 4/20 0.49
CDK8 P49336 1/20 0.49
KDR P35968 4/20 0.45
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 1/20 0.44
PIK3CG P48736 1/20 0.43
NR4A2 P43354 1/20 0.43
ATM Q13315 1/20 0.43
KDM5A P29375 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
NTRK1 P04629 1/20 0.42
PDGFRB P09619 1/20 0.42
KIT P10721 1/20 0.42
FLT3 P36888 1/20 0.42
MAP4K4 O95819 1/20 0.41
CRBN Q96SW2 1/20 0.40
CYP17A1 P05093 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3662014 0.92 FGFR3 (0.43) FGFR3FGFR1FYNCDK8KDR
SCHEMBL837839 0.82 FGFR1 (0.65) FGFR3FGFR1FYNCDK8HDAC8
SCHEMBL13336647 0.80 KDR (0.65) FGFR3FGFR1FYNKDRATM
SCHEMBL3030841 0.78 ATM (0.57) FGFR3FGFR1FYNKDRATM
Formic Acid SCHEMBL3318748 0.77 KDR (0.61) FGFR3FGFR1FYNKDRFLT3
SCHEMBL3033146 0.77 KDR (0.56) FGFR3FGFR1FYNKDRATM
SCHEMBL3031063 0.77 KDR (0.49) FGFR3FGFR1FYNKDRATM
SCHEMBL3025051 0.76 CDK8 (0.49) FGFR3FGFR1FYNCDK8KDR
SCHEMBL3029778 0.76 FGFR3 (0.50) FGFR3FGFR1FYNKDRATM
SCHEMBL3034200 0.76 FGFR3 (0.55) FGFR3FGFR1FYNKDRATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101827844-B Imidazo [1,2-a] pyridine derivatives useful as ALK inhibitors NOVARTIS AG 2013-08-14 CN disclosed
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
CN-101827844-A Imidazo [1,2-a] pyridine derivatives useful as ALK inhibitors NOVARTIS AG 2010-09-08 CN disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 FGFR3 32/4885FGFR1 72/4885FYN 1939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.