SCHEMBL30252597

SCHEMBL30252597

Nc1cc(-c2cnccn2)nc(-c2cnccn2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.44
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PI4KA P42356 1/20 0.42
PIK3CG P48736 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
HTT P42858 1/20 0.39
RECQL P46063 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GLA P06280 1/20 0.38
PIM1 P11309 4/20 0.38
NISCH Q9Y2I1 1/20 0.37
PIM2 Q9P1W9 2/20 0.36
CYP3A4 P08684 1/20 0.36
METAP2 P50579 1/20 0.36
ASIC3 Q9UHC3 1/20 0.35
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20911220 1.00 HSP90AA1 (0.44) HSP90AA1PIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL28996013 0.81 ASIC3 (0.52) HSP90AA1PIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL17755588 0.78 PIM1 (0.45) HTTRECQLPIM1NISCHCYP3A4
SCHEMBL29454745 0.78 NISCH (0.50) HSP90AA1HTTRECQLKDM4EPIM1
SCHEMBL78566 0.78 NISCH (0.50) HSP90AA1HTTRECQLKDM4EPIM1
SCHEMBL29598957 0.78 NISCH (0.50) HSP90AA1HTTRECQLKDM4EPIM1
SCHEMBL22334571 0.76 PIK3CD (0.45) HSP90AA1PIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL902145 0.76 KARS1 (0.44) HSP90AA1PIK3CDPIK3CAPIK3CBPI4KA
SCHEMBL31372462 0.75 NISCH (0.48) HSP90AA1HTTRECQLKDM4EPIM1
SCHEMBL14053846 0.75 NISCH (0.48) HSP90AA1HTTRECQLKDM4EPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651358-B 4-aminopyridine derivative, pharmaceutical composition, preparation method and application thereof 上海迪诺医药科技有限公司 2023-04-07 CN disclosed