SCHEMBL30253184

SCHEMBL30253184

COc1ccc2nc(SC(F)(F)F)sc2c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.70
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C19 P33261 2/20 0.55
APP P05067 2/20 0.55
PPARA Q07869 2/20 0.52
MAPT P10636 5/20 0.50
LMNA P02545 1/20 0.50
MAPK1 P28482 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TSHR P16473 1/20 0.49
HTT P42858 1/20 0.47
DYRK1A Q13627 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28589570 1.00 PDK1 (0.70) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL6693668 0.83 PDK1 (1.00) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL6902779 0.83 PDK1 (0.81) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL31291763 0.81 PDK1 (0.79) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL9389916 0.77 PDK1 (0.67) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL6692270 0.77 PDK1 (0.67) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL6691822 0.77 PDK1 (0.67) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL19435592 0.77 CYP1A2 (0.59) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL31294142 0.77 PDK1 (0.70) PDK1CYP1A2CYP3A4CYP2C19APP
SCHEMBL17950538 0.77 PDK1 (0.70) PDK1CYP1A2CYP3A4CYP2C19APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112939829-B Synthetic method of aryl trifluoromethyl thioether 武汉药明康德新药开发有限公司 2023-02-21 CN disclosed