SCHEMBL30253604

SCHEMBL30253604

c1ccc(-c2ccc3cc[nH]c3c2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.71
ADORA2A P29274 1/20 0.58
ADORA1 P30542 1/20 0.58
GHSR Q92847 2/20 0.56
AHR P35869 4/20 0.52
TRPA1 O75762 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
ITGB2 P05107 1/20 0.52
ICAM1 P05362 1/20 0.52
ITGAL P20701 1/20 0.52
CA4 P22748 1/20 0.52
CA6 P23280 1/20 0.52
ADK P55263 1/20 0.52
FGFR1 P11362 1/20 0.52
CMA1 P23946 1/20 0.50
TYR P14679 1/20 0.50
ENPP2 Q13822 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443799 1.00 NPC1 (0.71) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL7088159 0.96 NPC1 (0.67) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL7084471 0.86 NPC1 (0.58) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL7091322 0.86 NPC1 (0.54) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL446619 0.83 NPC1 (1.00) NPC1AHRTRPA1CA1CA2
SCHEMBL30587350 0.83 NPC1 (1.00) NPC1AHRTRPA1CA1CA2
Quinoline SCHEMBL27740778 0.83 NPC1 (0.51) NPC1ADORA2AADORA1GHSRAHR
Biphenyl SCHEMBL27962709 0.82 AHR (0.78) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL24601496 0.82 NPC1 (0.50) NPC1ADORA2AADORA1GHSRAHR
SCHEMBL1225643 0.82 TYR (0.70) NPC1AHRFGFR1CMA1TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4447954-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS Icahn School of Medicine at Mount Sinai (US) 2024-10-23 EP disclosed
CN-115806493-B Method for synthesizing epstein chiral intermediate by asymmetric hydrogenation 南京工业大学 2024-03-22 CN disclosed
WO-2023114472-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-22 WO disclosed
CN-115806493-A Method for synthesizing chiral ebavir intermediate by asymmetric hydrogenation 南京工业大学 2023-03-17 CN disclosed