SCHEMBL30254167

SCHEMBL30254167

C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCOCC5)nc(OCC56CCCN5CC(F)(F)C6)nc4c3F)c12

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.67
MAPK3 P27361 1/20 0.63
MAPK1 P28482 1/20 0.63
RAF1 P04049 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25081170 0.94 KRAS (0.66) KRASMAPK3MAPK1RAF1
SCHEMBL30254328 0.94 KRAS (0.66) KRASMAPK3MAPK1RAF1
SCHEMBL30254305 0.94 KRAS (0.66) KRASMAPK3MAPK1RAF1
SCHEMBL25081174 0.94 KRAS (0.66) KRASMAPK3MAPK1RAF1
SCHEMBL30254382 0.94 KRAS (0.66) KRASMAPK3MAPK1RAF1
SCHEMBL30254277 0.93 KRAS (0.76) KRASMAPK3MAPK1RAF1
SCHEMBL25080985 0.93 KRAS (0.76) KRASMAPK3MAPK1RAF1
SCHEMBL25081184 0.89 KRAS (0.83) KRASMAPK3MAPK1RAF1
SCHEMBL25080934 0.89 KRAS (0.83) KRASMAPK3MAPK1RAF1
SCHEMBL30254106 0.89 KRAS (0.83) KRASMAPK3MAPK1RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250019377-A1 1, 4-OXAZEPANE DERIVATIVES AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2025-01-16 US disclosed
EP-4387967-A1 1, 4-OXAZEPANE DERIVATIVES AND USES THEREOF Jacobio Pharmaceuticals Co., Ltd. (CN) 2024-06-26 EP disclosed
WO-2023020519-A9 1, 4-OXAZEPANE DERIVATIVES AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2023-03-23 WO disclosed
WO-2023020519-A1 1, 4-OXAZEPANE DERIVATIVES AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2023-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250019377-A1 1, 4-OXAZEPANE DERIVATIVES AND USES THEREOF CYP11B2, CYP21A2, CYP11B1 KRAS 2838/4885MAPK3 2751/4885MAPK1 2379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.