SCHEMBL3026751

SCHEMBL3026751

Fc1cccc(-c2ccn3c(-c4ccnc(-c5ccccc5F)c4)cnc3c2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.56
GABRB3 P28472 2/20 0.56
GABRA3 P34903 2/20 0.56
GABRA1 P14867 1/20 0.56
FLT3 P36888 7/20 0.54
KDR P35968 10/20 0.52
FGFR3 P22607 3/20 0.47
TGFBR1 P36897 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3026485 0.89 FLT3 (0.62) GABRG2GABRB3GABRA3FLT3KDR
SCHEMBL3032703 0.88 KDR (0.62) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3031225 0.86 GABRG2 (0.53) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3032514 0.84 GABRG2 (0.49) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3029113 0.84 GABRG2 (0.51) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3020791 0.83 KDR (0.50) GABRG2GABRB3GABRA3GABRA1KDR
SCHEMBL3033322 0.83 FLT3 (0.53) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3030180 0.83 GABRA1 (0.59) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3026843 0.83 GABRA1 (0.48) GABRG2GABRB3GABRA3GABRA1FLT3
SCHEMBL3028725 0.83 KDR (0.60) GABRG2GABRB3GABRA3FLT3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 GABRG2 2020/4885GABRB3 1344/4885GABRA3 1071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.