SCHEMBL30280409

SCHEMBL30280409

Ic1c[nH]c2ncccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.60
GPR84 Q9NQS5 1/20 0.58
LRRK2 Q5S007 1/20 0.55
KMT2A Q03164 1/20 0.55
CDC7 O00311 4/20 0.50
CDK2 P24941 3/20 0.50
MAP4K4 O95819 3/20 0.50
PIM1 P11309 3/20 0.50
PRKACA P17612 3/20 0.50
GSK3B P49841 3/20 0.50
HIPK2 Q9H2X6 3/20 0.50
CLK4 Q9HAZ1 3/20 0.50
MET P08581 2/20 0.50
ROCK2 O75116 2/20 0.50
IRAK4 Q9NWZ3 1/20 0.50
CAMKK2 Q96RR4 2/20 0.49
TGFBR1 P36897 3/20 0.49
PDPK1 O15530 2/20 0.49
IKBKE Q14164 2/20 0.49
MAP2K1 Q02750 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412615 1.00 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
Tert-Butyl Formate SCHEMBL27947847 0.82 KMT2A (0.50) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL5618155 0.78 TGFBR1 (0.71) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL2111969 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL368676 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL5802606 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL12605500 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL410624 0.75 AXL (1.00) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL12188 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7
SCHEMBL31097189 0.75 AXL (0.60) AXLGPR84LRRK2KMT2ACDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4522608-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2025-03-19 EP disclosed
CN-119546602-A Pyrrolidone derivatives as inhibitors of nfkb-induced kinase 詹森药业有限公司 2025-02-28 CN disclosed
CN-113874363-B Protein tyrosine phosphatase inhibitors ARRAY生物制药公司 2024-11-12 CN disclosed
WO-2023217906-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2023-11-16 WO disclosed
WO-2023064218-A1 TYRO3 INHIBITORS Halia Therapeutics, Inc. (US) 2023-04-20 WO disclosed