SCHEMBL30280762

SCHEMBL30280762

COC(=O)c1cc(C(=N)SC)cc(C2CCC2)c1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
HSP90AA1 P07900 2/20 0.32
HSP90AB1 P08238 2/20 0.32
OPRK1 P41145 2/20 0.32
LMNA P02545 2/20 0.30
POLB P06746 2/20 0.30
PTGER4 P35408 1/20 0.30
USP2 O75604 1/20 0.30
HSD17B10 Q99714 2/20 0.30
SLC6A3 Q01959 2/20 0.30
SCN9A Q15858 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
PDE5A O76074 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PRKCB P05771 1/20 0.30
PRKCA P17252 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30280863 0.85 DRD2 (0.32) PDK2PDK4ALDH1A1KDM4EOPRK1
SCHEMBL12488339 0.79 FASN (0.38) PDK2PDK4SLC6A3
SCHEMBL30281000 0.78 HSD17B10 (0.39) PDK2PDK4ALDH1A1KDM4EHSP90AA1
SCHEMBL30280829 0.77 ALDH1A1 (0.34) PDK2PDK4ALDH1A1KDM4EHSP90AA1
SCHEMBL30281011 0.76 OPRK1 (0.39) PDK2PDK4ALDH1A1KDM4EHSP90AA1
SCHEMBL12488689 0.75 MEN1 (0.33) PDK2PDK4ALDH1A1KDM4EOPRK1
SCHEMBL12488738 0.73 PDK2 (0.38) PDK2PDK4ALDH1A1KDM4ELMNA
SCHEMBL30280860 0.73 FASN (0.39) PDK2PDK4ALDH1A1KDM4EHSP90AA1
SCHEMBL12489060 0.73 PDK2 (0.38) PDK2PDK4ALDH1A1KDM4ELMNA
SCHEMBL30280814 0.72 FASN (0.40) PDK2PDK4OPRK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177551-B Heterocyclic modulators of lipid synthesis 3-V生物科学股份有限公司 2023-02-17 CN disclosed