SCHEMBL3029705

SCHEMBL3029705

c1cc(-c2cnc3cc(-c4ccncc4)ccn23)cc(-n2cccn2)c1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.65
FLT3 P36888 7/20 0.51
FGFR3 P22607 2/20 0.49
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA3 P34903 1/20 0.47
TBK1 Q9UHD2 1/20 0.45
PIK3CA P42336 1/20 0.42
MTOR P42345 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3022097 0.90 KDR (0.62) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3322220 0.90 FLT3 (0.66) KDRFLT3FGFR3
SCHEMBL3032319 0.84 FLT3 (0.53) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3031157 0.84 GABRG2 (0.52) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3021811 0.84 KDR (0.47) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3025334 0.84 KDR (0.47) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3026010 0.83 KDR (0.53) KDRFLT3FGFR3GABRG2GABRB3
SCHEMBL3025677 0.82 KDR (0.48) KDRFGFR3GABRG2GABRB3GABRA3
SCHEMBL3029778 0.80 FGFR3 (0.50) KDRFLT3FGFR3TBK1
SCHEMBL5248501 0.80 KDR (1.00) KDRFLT3FGFR3GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP claimed
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
EP-2212323-B1 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2012-08-15 EP disclosed
US-20100210641-A1 Organic Compounds NOVARTIS AG (CH) 2010-08-19 US disclosed
EP-2212323-A2 IMIDAZO [1,2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS Novartis AG (CH) 2010-08-04 EP disclosed
WO-2009050183-A2 IMIDAZO [1, 2-A] PYRIDINE DERIVATIVES USEFUL AS ALK INHIBITORS NOVARTIS AG (CH) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210641-A1 Organic Compounds ALK, ACVR1, ACVRL1 KDR 372/4885FLT3 4384/4885FGFR3 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.