Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | KDM4E | B2RXH2 | 5/20 | 0.46 |
| ▸ | GPR3 | P46089 | 1/20 | 0.46 |
| ▸ | MAPT | P10636 | 3/20 | 0.39 |
| ▸ | CASP3 | P42574 | 1/20 | 0.39 |
| ▸ | SMN1; SMN2 | Q16637 | 3/20 | 0.38 |
| ▸ | ALOX15 | P16050 | 2/20 | 0.38 |
| ▸ | PDPK1 | O15530 | 1/20 | 0.38 |
| ▸ | CA12 | O43570 | 1/20 | 0.38 |
| ▸ | PARP1 | P09874 | 1/20 | 0.38 |
| ▸ | CA9 | Q16790 | 1/20 | 0.38 |
| ▸ | TNKS2 | Q9H2K2 | 1/20 | 0.38 |
| ▸ | ERN1 | O75460 | 1/20 | 0.38 |
| ▸ | HSD17B10 | Q99714 | 3/20 | 0.36 |
| ▸ | HPGD | P15428 | 2/20 | 0.36 |
| ▸ | ALDH1A1 | P00352 | 3/20 | 0.35 |
| ▸ | CDK4 | P11802 | 1/20 | 0.35 |
| ▸ | CCND1 | P24385 | 1/20 | 0.35 |
| ▸ | HTT | P42858 | 1/20 | 0.35 |
| ▸ | NPSR1 | Q6W5P4 | 1/20 | 0.35 |
| ▸ | MAOA | P21397 | 2/20 | 0.35 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL31672121 | 0.78 | KDM4E (0.38) | KDM4EGPR3MAPTCASP3SMN1; SMN2 | |
| SCHEMBL1920170 | 0.72 | CA12 (0.42) | KDM4EGPR3SMN1; SMN2ALOX15PDPK1 | |
| SCHEMBL30617063 | 0.72 | DNMT1 (0.44) | KDM4EMAPTHSD17B10HPGDALDH1A1 | |
| SCHEMBL6759607 | 0.72 | DNMT1 (0.44) | KDM4EMAPTHSD17B10HPGDALDH1A1 | |
| SCHEMBL16352244 | 0.70 | MAOA (0.52) | KDM4EGPR3MAPTSMN1; SMN2HSD17B10 | |
| SCHEMBL16836537 | 0.69 | KDM4E (0.39) | KDM4EGPR3MAPTCASP3SMN1; SMN2 | |
| SCHEMBL31475620 | 0.69 | MAOA (0.46) | KDM4EMAPTCASP3SMN1; SMN2ALOX15 | |
| SCHEMBL28922775 | 0.69 | MAOA (0.46) | KDM4EMAPTCASP3SMN1; SMN2ALOX15 | |
| SCHEMBL28480419 | 0.68 | HPRT1 (0.50) | HSD17B10HPGDALDH1A1TDP1USP2 | |
| SCHEMBL7818325 | 0.68 | KDM4E (0.41) | KDM4EGPR3MAPTSMN1; SMN2ERN1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20230075190-A1 | COMPOSITIONS AND METHODS OF USE THEREOF FOR TREATMENT OR PREVENTION OF CONDITIONS ASSOCIATED WITH HYPERPROLIFERATIVE CELLULAR DIVISION, DIABETES, IMMUNODEFICIENCY DISEASES, ALZHEIMER'S DISEASE OR AUTOIMMUNE DISEASES, AND TESTING SYSTEM AND METHOD | CHAI FOUNDATION FOR MEDICAL RES & LIFE EXTENSION INC (US) | 2023-03-09 | — | — | US | claimed |
| US-20240052418-A1 | METHOD FOR PREDICTING A SUBJECT'S RESPONSE TO SLC MODULATOR THERAPY | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2024-02-15 | — | — | US | disclosed |
| US-11814681-B2 | Method for predicting a subjects response to SLC modulator therapy | THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) | 2023-11-14 | — | — | US | disclosed |
| US-20230075190-A1 | COMPOSITIONS AND METHODS OF USE THEREOF FOR TREATMENT OR PREVENTION OF CONDITIONS ASSOCIATED WITH HYPERPROLIFERATIVE CELLULAR DIVISION, DIABETES, IMMUNODEFICIENCY DISEASES, ALZHEIMER'S DISEASE OR AUTOIMMUNE DISEASES, AND TESTING SYSTEM AND METHOD | CHAI FOUNDATION FOR MEDICAL RES & LIFE EXTENSION INC (US) | 2023-03-09 | — | — | US | disclosed |