SCHEMBL30301447

SCHEMBL30301447

COc1ccc(CN(C[C@H](C)O)C(=O)c2n[nH]c3nc(Cl)ccc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PSEN1 P49768 1/20 0.35
PSEN2 P49810 1/20 0.35
APH1B Q8WW43 1/20 0.35
NCSTN Q92542 1/20 0.35
APH1A Q96BI3 1/20 0.35
PSENEN Q9NZ42 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
USP2 O75604 2/20 0.35
TUBB4A P04350 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30301453 0.79 PRKACA (0.44) ALDH1A1NPSR1TSHRPRKACAPRKACG
SCHEMBL23160276 0.79 TSHR (0.46) ALDH1A1NPSR1TDP1TSHRPSEN1
SCHEMBL29731691 0.79 TSHR (0.46) ALDH1A1NPSR1TDP1TSHRPSEN1
SCHEMBL30301483 0.72 GAA (0.38) ALDH1A1NPSR1HTTSMN1; SMN2
SCHEMBL20472046 0.71 ALDH1A1 (0.52) ALDH1A1NPSR1TDP1TSHRUSP2
SCHEMBL29863299 0.69 POLB (0.41) ALDH1A1NPSR1TDP1TSHRPRKACA
SCHEMBL22413013 0.69 POLB (0.41) ALDH1A1NPSR1TDP1TSHRPRKACA
SCHEMBL16532656 0.69 KDM4E (0.53) ALDH1A1NPSR1TUBB4ATUBBTUBA3C
SCHEMBL18179687 0.68 ACR (0.51) ALDH1A1HTTSMN1; SMN2
SCHEMBL24610141 0.65 ALDH1A1 (0.43) ALDH1A1NPSR1TDP1TSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023025109-A1 TOLL-LIKE RECEPTOR INHIBITOR AND PREPARATION AND APPLICATION THEREOF 上海维申医药有限公司 2023-03-02 WO disclosed