SCHEMBL30309486

SCHEMBL30309486

COc1ccc(N2C(=O)N(c3c(CF)csc3Cl)Cc3cnc(Cl)nc32)nc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIK2 Q9H0K1 2/20 0.46
CSF1R P07333 1/20 0.43
SIK1 P57059 1/20 0.43
SIK3 Q9Y2K2 1/20 0.43
FGFR4 P22455 15/20 0.33
FGFR1 P11362 11/20 0.33
FGFR2 P21802 6/20 0.32
FGFR3 P22607 5/20 0.32
KDR P35968 1/20 0.32
LCK P06239 1/20 0.31
MAPK14 Q16539 1/20 0.31
DHFR P00374 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25882416 1.00 SIK2 (0.46) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL23978369 0.90 FGFR4 (0.40) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309508 0.90 FGFR4 (0.40) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309533 0.88 SIK2 (0.51) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL23978120 0.88 SIK2 (0.51) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309495 0.86 SIK2 (0.47) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309484 0.82 SIK2 (0.71) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL25881931 0.81 CSF1R (0.60) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309616 0.81 CSF1R (0.60) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309527 0.81 SIK2 (0.53) SIK2CSF1RSIK1SIK3FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143191-A2 BICYCLIC KINASE INHIBITORS AND USES THEREOF iOmx Therapeutics AG (DE) 2023-03-08 EP disclosed