SCHEMBL30309533

SCHEMBL30309533

COc1ccc(N2C(=O)N(c3c(C)csc3Cl)Cc3cnc(Cl)nc32)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIK2 Q9H0K1 2/20 0.51
CSF1R P07333 1/20 0.48
SIK1 P57059 1/20 0.48
SIK3 Q9Y2K2 1/20 0.48
FGFR4 P22455 14/20 0.34
FGFR1 P11362 13/20 0.34
FGFR2 P21802 6/20 0.33
FGFR3 P22607 5/20 0.33
KDR P35968 1/20 0.33
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31
TUBB8 Q3ZCM7 1/20 0.31
TUBA3E Q6PEY2 1/20 0.31
TUBA1A Q71U36 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978120 1.00 SIK2 (0.51) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309486 0.88 SIK2 (0.46) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL25882416 0.88 SIK2 (0.46) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309495 0.88 SIK2 (0.47) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL23978372 0.85 SIK2 (0.68) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309504 0.85 SIK2 (0.68) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309511 0.83 SIK2 (0.51) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL23978178 0.83 SIK2 (0.51) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL30309560 0.83 SIK2 (0.49) SIK2CSF1RSIK1SIK3FGFR4
SCHEMBL25882388 0.83 SIK2 (0.49) SIK2CSF1RSIK1SIK3FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4143191-A2 BICYCLIC KINASE INHIBITORS AND USES THEREOF iOmx Therapeutics AG (DE) 2023-03-08 EP disclosed