SCHEMBL30320141

SCHEMBL30320141

COCCOc1cccc(CCN2C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.53
PKM P14618 1/20 0.48
PDE10A Q9Y233 1/20 0.46
ALDH1A1 P00352 3/20 0.45
POLB P06746 2/20 0.45
RAB9A P51151 5/20 0.45
MAPT P10636 4/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
LMNA P02545 3/20 0.44
HPGD P15428 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 1/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24618502 1.00 HSD17B10 (0.53) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL17391050 0.85 HSD17B10 (0.56) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL30320202 0.85 HSD17B10 (0.56) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL9447444 0.76 PKM (0.61) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL30320196 0.74 HRH1 (0.41) TSHRCYP2C9CYP2C19
SCHEMBL24618504 0.74 HRH1 (0.41) TSHRCYP2C9CYP2C19
SCHEMBL3642366 0.73 RAB9A (0.65) ALDH1A1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL29530672 0.73 RAB9A (0.65) ALDH1A1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL5348595 0.73 HSD17B10 (0.60) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL2210883 0.72 RAB9A (0.72) HSD17B10ALDH1A1POLBRAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867553-A Diaminopyrazolo [1,5-a ] pyrimidine-6-carbonitrile compounds as adenosine 2A receptor and adenosine 2B receptor antagonists 巴格沃克斯研究有限公司 2023-03-28 CN disclosed