SCHEMBL30320202

SCHEMBL30320202

COc1cccc(CCN2C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.56
PKM P14618 1/20 0.53
PDE10A Q9Y233 2/20 0.51
ALDH1A1 P00352 4/20 0.50
POLB P06746 2/20 0.50
MAPT P10636 3/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
LMNA P02545 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 2/20 0.46
MAPK1 P28482 1/20 0.46
GLS O94925 1/20 0.45
RXFP1 Q9HBX9 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
HPGD P15428 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
GAA P10253 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17391050 1.00 HSD17B10 (0.56) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL24618502 0.85 HSD17B10 (0.53) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL30320141 0.85 HSD17B10 (0.53) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL9447444 0.81 PKM (0.61) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL5348595 0.78 HSD17B10 (0.60) HSD17B10PKMPDE10AALDH1A1POLB
SCHEMBL27366781 0.78 MTNR1A (0.53) PDE10AALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL31332177 0.78 MTNR1A (0.53) PDE10AALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL20796153 0.75 PGK1 (0.44) HSD17B10PDE10AALDH1A1MAPTMEN1
SCHEMBL29828797 0.73 KDM4E (0.53) HSD17B10PKMALDH1A1MAPTLMNA
SCHEMBL27032749 0.73 KDM4E (0.53) HSD17B10PKMALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867553-A Diaminopyrazolo [1,5-a ] pyrimidine-6-carbonitrile compounds as adenosine 2A receptor and adenosine 2B receptor antagonists 巴格沃克斯研究有限公司 2023-03-28 CN disclosed