SCHEMBL30323

SCHEMBL30323

O=C(Nc1nc2ccc(O)cc2s1)c1cccc(O)c1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 9/20 1.00
HSD17B2 P37059 8/20 1.00
CYP3A4 P08684 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2B6 P20813 1/20 0.68
CYP2C19 P33261 1/20 0.68
DYRK1A Q13627 3/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
DYRK1B Q9Y463 2/20 0.57
DYRK2 Q92630 1/20 0.55
SNCA P37840 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29870 0.86 HSD17B1 (0.75) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29886 0.83 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29710 0.83 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL31033 0.82 HSD17B1 (0.76) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL31050 0.81 HSD17B1 (0.68) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL29964 0.81 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL13329184 0.80 HSD17B1 (0.81) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL13329867 0.80 HSD17B1 (0.66) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL12199345 0.80 HSD17B1 (0.66) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9
SCHEMBL12199320 0.80 HSD17B1 (0.81) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed