SCHEMBL30353086

SCHEMBL30353086

Cn1nc(-c2ccccc2)cc1Oc1cc(C#N)ccc1-c1ccc(CCN)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.40
CYP19A1 P11511 3/20 0.40
CYP11B2 P19099 2/20 0.40
SCN9A Q15858 1/20 0.39
PIN1 Q13526 1/20 0.36
PHGDH O43175 1/20 0.35
NSD2 O96028 2/20 0.34
GRM5 P41594 1/20 0.34
ADRA2C P18825 1/20 0.34
ALOX5AP P20292 2/20 0.33
FEN1 P39748 1/20 0.33
KDM1A O60341 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
SQOR Q9Y6N5 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
GABRG2 P18507 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25554071 1.00 CYP11B1 (0.40) CYP11B1CYP19A1CYP11B2SCN9APIN1
SCHEMBL25554271 0.93 SCN9A (0.40) CYP11B1CYP19A1CYP11B2SCN9APIN1
SCHEMBL30353051 0.93 SCN9A (0.40) CYP11B1CYP19A1CYP11B2SCN9APIN1
SCHEMBL25554077 0.92 CYP11B2 (0.47) CYP11B1CYP19A1CYP11B2SCN9AKDM4E
SCHEMBL25554088 0.92 NSD2 (0.37) CYP11B1CYP19A1CYP11B2SCN9ANSD2
SCHEMBL30353115 0.92 NSD2 (0.37) CYP11B1CYP19A1CYP11B2SCN9ANSD2
SCHEMBL30353104 0.92 GRM5 (0.38) CYP11B1CYP19A1CYP11B2SCN9ANSD2
SCHEMBL25554119 0.92 GRM5 (0.38) CYP11B1CYP19A1CYP11B2SCN9ANSD2
SCHEMBL25554706 0.90 CYP11B1 (0.36) CYP11B1CYP19A1CYP11B2SCN9ANSD2
SCHEMBL25554247 0.90 CYP11B1 (0.41) CYP11B1CYP19A1CYP11B2SCN9APIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN claimed
CN-115996910-A Aryl or heteroaryl derivatives 帝人制药株式会社 2023-04-21 CN disclosed