SCHEMBL3035529

SCHEMBL3035529

CC(C)N1CCN(c2cncc(-c3ccccc3)c2)CC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.52
CHRNA3 P32297 1/20 0.52
VCP P55072 1/20 0.45
KHK P50053 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
TGFBR1 P36897 1/20 0.44
ACVR1 Q04771 1/20 0.44
KCNH2 Q12809 1/20 0.44
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
CHEK1 O14757 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
MCOLN2 Q8IZK6 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3453906 0.83 CHEK1 (0.58) CHRNB4CHRNA3ACVR1CHEK1
SCHEMBL13778275 0.78 TGFBR1 (0.54) KHKKDM4EALDH1A1MAPTPKM
SCHEMBL6357589 0.78 CHEK1 (0.53) CHRNB4CHRNA3ACVR1CHEK1
SCHEMBL3453352 0.77 HTR1A (0.66) CHRNB4CHRNA3TGFBR1
SCHEMBL27818822 0.77 CHRNB4 (0.52) CHRNB4CHRNA3ALDH1A1MAPTDRD2
SCHEMBL15345003 0.76 KDM4E (0.46) CHRNB4CHRNA3KHKKDM4EALDH1A1
Hydrochloric Acid SCHEMBL3268024 0.76 HTR1A (0.64) CHRNB4CHRNA3TGFBR1ACVR1
SCHEMBL12321710 0.75 CHRNB2 (0.55) CHRNB4CHRNA3VCPKHKKDM4E
SCHEMBL12326041 0.75 KDM4E (0.45) VCPKHKKDM4EALDH1A1MAPT
SCHEMBL13436330 0.75 KDM4E (0.45) VCPKHKKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233470-A1 Histamine H3 receptor antagonists High Point Pharmaceuticals, LLC (US) 2010-09-29 EP disclosed