SCHEMBL30358192

SCHEMBL30358192

O=C(Oc1ccc2c(ccc3ccccc32)c1)c1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.78
MAPT P10636 5/20 0.78
TDP1 Q9NUW8 2/20 0.78
MEN1 O00255 2/20 0.78
CA9 Q16790 3/20 0.57
CA12 O43570 2/20 0.57
POLB P06746 1/20 0.55
PDGFRB P09619 2/20 0.53
PDGFRA P16234 2/20 0.53
ALDH1A1 P00352 4/20 0.50
PARP10 Q53GL7 1/20 0.50
HPGD P15428 1/20 0.50
KDM4E B2RXH2 1/20 0.50
GLA P06280 1/20 0.50
GAA P10253 1/20 0.50
NPBWR1 P48145 1/20 0.50
HSD17B10 Q99714 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
PKM P14618 1/20 0.47
PTGES O14684 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27945114 0.92 KMT2A (0.71) KMT2AMAPTTDP1MEN1CA9
SCHEMBL31365678 0.92 KMT2A (0.75) KMT2AMAPTTDP1MEN1CA9
SCHEMBL27858102 0.92 KMT2A (0.75) KMT2AMAPTTDP1MEN1CA9
SCHEMBL1639878 0.88 KMT2A (1.00) KMT2AMAPTTDP1MEN1CA9
SCHEMBL30523105 0.88 KMT2A (1.00) KMT2AMAPTTDP1MEN1CA9
Ammonia Solution, Strong SCHEMBL11705203 0.86 KMT2A (0.96) KMT2AMAPTTDP1MEN1CA9
SCHEMBL18058690 0.84 KMT2A (0.93) KMT2AMAPTTDP1MEN1CA9
SCHEMBL31499302 0.84 KMT2A (0.56) KMT2AMAPTTDP1MEN1CA9
Benzoic Acid SCHEMBL9956914 0.83 KMT2A (0.90) KMT2AMAPTTDP1MEN1CA9
SCHEMBL27267214 0.82 ALOX5 (0.60) KMT2AMAPTTDP1MEN1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118724999-A Synthesis of cholic acid derivative and application of cholic acid derivative as TGR5 allosteric agonist 常州大学 2024-10-01 CN disclosed
CN-115710298-B Cholic acid derivative, preparation method thereof and application of cholic acid derivative as TGR5 allosteric agonist 常州大学 2024-10-01 CN disclosed
WO-2023168974-A1 CHOLIC ACID DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF AS TGR5 ALLOSTERIC AGONIST 常州大学 2023-09-14 WO disclosed
CN-115943307-A MR1 ligands and pharmaceutical compositions for immunomodulation 巴塞尔大学 2023-04-07 CN disclosed