SCHEMBL30359003

SCHEMBL30359003

COc1ccc(C)c(C(=O)N2C3CNCC2CC(=O)C3)n1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 3/20 0.42
CHRNA4 P43681 3/20 0.36
KCNK3 O14649 8/20 0.35
KCNK9 Q9NPC2 8/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
HCRTR1 O43613 3/20 0.33
HCRTR2 O43614 3/20 0.33
NNMT P40261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30359044 0.89 HTR2A (0.41) HTR2AHTR2CHTR2BCHRNA4KCNK3
SCHEMBL30359111 0.89 HTR2A (0.41) HTR2AHTR2CHTR2BCHRNA4KCNK3
SCHEMBL30359053 0.87 KCNK3 (0.42) HTR2AHTR2CHTR2BKCNK3KCNK9
SCHEMBL30359037 0.80 KCNK3 (0.41) HTR2AHTR2CHTR2BKCNK3KCNK9
SCHEMBL30359162 0.80 MGLL (0.43) HTR2AHTR2CHTR2BKCNK3KCNK9
SCHEMBL30359062 0.76 KCNK3 (0.48) HTR2AHTR2CHTR2BKCNK3KCNK9
SCHEMBL30359131 0.76 KCNK3 (0.47) HTR2AHTR2CHTR2BKCNK3KCNK9
SCHEMBL20587387 0.72 KCNK3 (0.46) KCNK3KCNK9HCRTR1HCRTR2
SCHEMBL21904724 0.72 KCNK3 (0.45) KCNK3KCNK9
SCHEMBL30359095 0.72 KCNK3 (0.46) KCNK3KCNK9HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116057057-A Conjugates of alpha 2-adrenoceptor subtype C (alpha-2C) antagonists and TASK1/3 channel blockers for the treatment of sleep apnea 拜耳公司 2023-05-02 CN disclosed