SCHEMBL30359409

SCHEMBL30359409

NC(=O)c1cccnc1OCC1CC1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.51
RAB9A P51151 1/20 0.50
PARP10 Q53GL7 6/20 0.49
PARP15 Q460N3 5/20 0.49
PARP2 Q9UGN5 2/20 0.49
PARP1 P09874 1/20 0.47
IRAK4 Q9NWZ3 5/20 0.47
ROCK2 O75116 4/20 0.46
FFAR4 Q5NUL3 1/20 0.43
GRM4 Q14833 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5955514 1.00 ACHE (0.51) ACHERAB9APARP10PARP15PARP2
SCHEMBL30314024 0.90 IRAK4 (0.56) ACHERAB9AIRAK4GRM4
SCHEMBL14334795 0.90 IRAK4 (0.56) ACHERAB9AIRAK4GRM4
SCHEMBL14334981 0.90 IRAK4 (0.49) ACHERAB9APARP1IRAK4ROCK2
SCHEMBL14334294 0.86 IRAK4 (0.60) ACHEPARP1IRAK4ROCK2
SCHEMBL14334551 0.83 IRAK4 (0.59) PARP1IRAK4ROCK2
SCHEMBL19149183 0.81 ROCK2 (0.48) RAB9APARP10PARP15PARP1ROCK2
SCHEMBL3669098 0.80 IRAK4 (0.58) RAB9APARP1IRAK4ROCK2GRM4
SCHEMBL23462725 0.80 ROCK2 (0.53) ACHEIRAK4ROCK2
SCHEMBL14335146 0.80 CYP4F2 (0.49) ACHEIRAK4ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12509424-B2 Compound and composition as PDGF receptor kinase inhibitor NIPPON SHINYAKU CO., LTD. (JP) 2025-12-30 US disclosed
US-20230101484-A1 COMPOUND AND COMPOSITION AS PDGF RECEPTOR KINASE INHIBITOR NIPPON SHINYAKU CO., LTD. (JP) 2023-03-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12509424-B2 Compound and composition as PDGF receptor kinase inhibitor PDGFRA, PDGFRB, PDGFA ACHE 4635/4885RAB9A 2815/4885PARP10 1716/4885
US-20230101484-A1 COMPOUND AND COMPOSITION AS PDGF RECEPTOR KINASE INHIBITOR PDGFRB, PDGFRA, PDGFA ACHE 4538/4885RAB9A 2531/4885PARP10 1465/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.