SCHEMBL30362298

SCHEMBL30362298

CCc1nn(-c2ccc(NC(=O)OC(C)(C)C)cn2)cc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 7/20 0.36
AAK1 Q2M2I8 2/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
MAPK14 Q16539 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
NAMPT P43490 1/20 0.34
SCD O00767 1/20 0.34
CYP17A1 P05093 1/20 0.33
GSK3B P49841 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25254861 1.00 MAPKAPK2 (0.36) MAPKAPK2AAK1PRMT5WDR77PTGDR2
SCHEMBL25251320 0.88 PTGDR2 (0.38) MAPKAPK2AAK1PRMT5WDR77PTGDR2
SCHEMBL30362248 0.88 PTGDR2 (0.38) MAPKAPK2AAK1PRMT5WDR77PTGDR2
SCHEMBL25352595 0.88 UCHL1 (0.36)
SCHEMBL30362262 0.86 NAMPT (0.35) MAPKAPK2AAK1PRMT5WDR77PTGDR2
SCHEMBL25350925 0.86 NAMPT (0.35) MAPKAPK2AAK1PRMT5WDR77PTGDR2
SCHEMBL30362342 0.85 AR (0.39) MAPKAPK2AAK1NAMPT
SCHEMBL25297826 0.85 AR (0.39) MAPKAPK2AAK1NAMPT
SCHEMBL25253508 0.81 MAPKAPK2 (0.41) MAPKAPK2PTGDR2MAPK14HDAC3HDAC8
SCHEMBL29004191 0.80 FFAR1 (0.41) MAPKAPK2AAK1PRMT5WDR77HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115989225-A Imidazole-pyrazole derivatives as antibacterial agents 豪夫迈·罗氏有限公司 2023-04-18 CN disclosed