SCHEMBL30366148

SCHEMBL30366148

Cc1c(C(N)=O)sc2nccn12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
GRM5 P41594 1/20 0.42
LIMK1 P53667 4/20 0.40
IKBKB O14920 6/20 0.38
CHUK O15111 1/20 0.38
IDO1 P14902 1/20 0.37
CHRM4 P08173 2/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
ZAP70 P43403 1/20 0.35
SYK P43405 1/20 0.35
KARS1 Q15046 1/20 0.35
CDC7 O00311 1/20 0.35
DBF4 Q9UBU7 1/20 0.35
CDK8 P49336 2/20 0.34
DAPK3 O43293 1/20 0.34
PRKD3 O94806 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL275781 0.84 GRM5 (0.43) MAPTNPC1RAB9AGRM5IDO1
SCHEMBL275779 0.79 GRM5 (0.43) MAPTNPC1RAB9AGRM5ALDH1A1
SCHEMBL3459509 0.72 IDO1 (0.51) GRM5LIMK1IDO1CHRM4CDK8
SCHEMBL19830990 0.70 CHRM4 (0.70) LIMK1IKBKBCHUKCHRM4CDK8
SCHEMBL8054669 0.69 MAPT (0.43) MAPTNPC1RAB9AIKBKBIDO1
SCHEMBL4016458 0.67 IDO1 (0.39) NPC1RAB9AGRM5IDO1ALDH1A1
SCHEMBL4016456 0.67 IDO1 (0.39) GRM5IDO1
SCHEMBL28888466 0.66 IKBKB (0.38) MAPTNPC1RAB9ALIMK1IKBKB
SCHEMBL30085742 0.64 ADORA3 (0.36) LIMK1CHRM4CDK8DAPK3PRKD3
SCHEMBL284637 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789648-A Nitrile-containing antiviral compounds 辉瑞大药厂 2023-09-22 CN disclosed
CN-114466838-B Nitrile-containing antiviral compounds 辉瑞大药厂 2023-05-02 CN disclosed