SCHEMBL30367018

SCHEMBL30367018

Cc1ccnc(Oc2ccc(-c3c(Br)n(C)c4c(C#N)cnc(N)c34)cc2F)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
FGFR1 P11362 1/20 0.46
CYP2C9 P11712 1/20 0.46
FGFR2 P21802 1/20 0.46
FGFR4 P22455 1/20 0.46
FGFR3 P22607 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX5AP P20292 9/20 0.43
FEN1 P39748 9/20 0.43
KDM4E B2RXH2 1/20 0.35
KDM1A O60341 4/20 0.34
PI4KB Q9UBF8 1/20 0.33
GRM2 Q14416 1/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30366660 0.87 TNK2 (0.34) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL30367019 0.84 ALOX5AP (0.48) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL31361305 0.81 CYP2C9 (0.45) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL30848700 0.81 CYP3A4 (0.47) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL28981114 0.80 FGFR1 (0.65) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL30325867 0.80 FGFR1 (0.65) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL31213850 0.80 FGFR1 (0.73) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL31213925 0.80 FGFR4 (0.60) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL30325667 0.80 CYP3A4 (0.64) CYP3A4CYP2D6FGFR1CYP2C9FGFR2
SCHEMBL30366887 0.79 CYP3A4 (0.41) CYP3A4CYP2D6FGFR1CYP2C9FGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed