SCHEMBL30367405

SCHEMBL30367405

CCn1nc(N)c2c(-c3ccc(N)cc3)cc(C3=CCN(C(=O)C(C)C)CC3)cc21

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 11/20 0.41
KHK P50053 1/20 0.36
QDPR P09417 2/20 0.35
CCR1 P32246 1/20 0.35
CNR1 P21554 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
BTK Q06187 1/20 0.33
NPC1 O15118 1/20 0.33
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30367031 0.89 NAMPT (0.43) NAMPTKHKQDPRCCR1CNR1
SCHEMBL30367296 0.79 MAPK1 (0.39) NAMPTCCR1BTK
SCHEMBL30367298 0.72 NAMPT (0.48) NAMPTQDPRCCR1KCNH2HRH3
SCHEMBL30367241 0.70 NAMPT (0.43) NAMPTQDPRCCR1KCNH2HRH3
SCHEMBL29052499 0.70 NAMPT (0.40) NAMPTQDPRBTK
SCHEMBL30367401 0.69 NAMPT (0.36) NAMPT
SCHEMBL30585453 0.68 LYN (0.43) NAMPT
SCHEMBL30367181 0.68 LMNA (0.37)
SCHEMBL14197130 0.68 NAMPT (0.58) NAMPTQDPRCCR1KCNH2HRH3
SCHEMBL30367384 0.67 MAPK1 (0.40) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023155886-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-08-24 WO disclosed
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed
WO-2023051464-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-04-06 WO disclosed