SCHEMBL30367688

SCHEMBL30367688

CC(C)C(=O)N1CCC(c2cc(-c3ccc(NC(=O)c4cncc(-c5ccc(F)cc5)c4O)cc3)c3c(N)nn(C)c3c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MERTK Q12866 9/20 0.46
TYRO3 Q06418 9/20 0.45
KDR P35968 3/20 0.42
DYRK3 O43781 3/20 0.42
ROCK2 O75116 3/20 0.42
MAP4K4 O95819 3/20 0.42
CSF1R P07333 3/20 0.42
LYN P07948 3/20 0.42
RET P07949 3/20 0.42
MET P08581 3/20 0.42
KIT P10721 3/20 0.42
FGFR1 P11362 3/20 0.42
FLT1 P17948 3/20 0.42
RPS6KB1 P23443 3/20 0.42
EPHA2 P29317 3/20 0.42
FLT4 P35916 3/20 0.42
FRK P42685 3/20 0.42
CSNK1A1 P48729 3/20 0.42
CSNK1D P48730 3/20 0.42
CLK2 P49760 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29052756 1.00 MERTK (0.46) MERTKTYRO3KDRDYRK3ROCK2
SCHEMBL29052490 0.87 MET (0.51) MERTKTYRO3METAXL
SCHEMBL30367687 0.87 MET (0.51) MERTKTYRO3METAXL
SCHEMBL29052441 0.86 MERTK (0.46) MERTKTYRO3KDRCSF1RLYN
SCHEMBL30367348 0.86 MERTK (0.46) MERTKTYRO3KDRCSF1RLYN
SCHEMBL30367626 0.84 TYRO3 (0.55) MERTKTYRO3AXL
SCHEMBL29052459 0.84 TYRO3 (0.55) MERTKTYRO3AXL
SCHEMBL30367373 0.82 TYRO3 (0.47) MERTKTYRO3AXL
SCHEMBL30367283 0.81 MERTK (0.46) MERTKTYRO3KDR
SCHEMBL30367384 0.79 MAPK1 (0.40) MERTKTYRO3KDRDYRK3ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023155886-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-08-24 WO disclosed
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed
WO-2023051464-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-04-06 WO disclosed