SCHEMBL30397908

SCHEMBL30397908

COc1nc(NN)ncc1C#N

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
IDH1 O75874 15/20 0.44
IDH2 P48735 1/20 0.42
KCNH2 Q12809 1/20 0.42
MAPT P10636 1/20 0.41
LRRK2 Q5S007 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25226820 1.00 GAA (0.47) GAAKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL25597187 0.85 IDH1 (0.45) GAAIDH1IDH2KCNH2LRRK2
SCHEMBL26977882 0.77 ADORA2A (0.47) GAAKDM4EALDH1A1L3MBTL1MAPT
SCHEMBL9393281 0.75 KMT2A (0.46) GAAKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL21550205 0.75 GAA (0.44) GAAKDM4EALDH1A1L3MBTL1IDH1
SCHEMBL3817806 0.75 KDM4E (0.42) GAAKDM4EALDH1A1L3MBTL1IDH1
SCHEMBL25678881 0.75 CTSK (0.50) GAAKDM4EALDH1A1IDH1LRRK2
SCHEMBL5764208 0.75 KDM4E (0.48) GAAKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL20836481 0.74 ULK1 (0.47) GAAKDM4EALDH1A1LMNAL3MBTL1
SCHEMBL2527306 0.74 PIN1 (0.59) GAAKDM4EALDH1A1L3MBTL1IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed